GABRA1 (GABA-A Receptor)

GABRA1

Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.

機能

Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.

この標的に作用する薬物

薬物 作用 主要
Diazepam Agonist はい
Alprazolam Agonist はい
Zolpidem Agonist はい
Memantine Antagonist はい
Valproic Acid Agonist
Topiramate Agonist

Related Targets