GABRA1 (GABA-A Receptor)

GABRA1

Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.

Function

Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.

Drugs Acting on This Target

Drug Action Primary
Diazepam Agonist Yes
Zolpidem Agonist Yes
Alprazolam Agonist Yes

Related Targets