SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
機能
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
この標的に作用する薬物
| 薬物 | 作用 | 主要 |
|---|---|---|
| Valproic Acid | Blocker | はい |
| Topiramate | Blocker | はい |
| Phenytoin | Blocker | はい |
| Gabapentin | Blocker | はい |
| Pregabalin | Blocker | はい |
| Lamotrigine | Blocker | はい |
| Carbamazepine | Blocker | はい |
| Furosemide | Inhibitor | はい |
| Hydrochlorothiazide | Inhibitor | はい |