GABRA1 (GABA-A Receptor)
GABRA1
Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.
Fonction
Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.
Médicaments agissant sur cette cible
| Médicament | Action | Principal |
|---|---|---|
| Diazepam | Agonist | Oui |
| Alprazolam | Agonist | Oui |
| Zolpidem | Agonist | Oui |
| Memantine | Antagonist | Oui |
| Valproic Acid | Agonist | — |
| Topiramate | Agonist | — |