GABRA1 (GABA-A Receptor)
GABRA1
Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.
İşlev
Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.
Bu Hedefe Etki Eden İlaçlar
| İlaç | Etki | Birincil |
|---|---|---|
| Diazepam | Agonist | Evet |
| Alprazolam | Agonist | Evet |
| Zolpidem | Agonist | Evet |
| Memantine | Antagonist | Evet |
| Valproic Acid | Agonist | — |
| Topiramate | Agonist | — |