GABRA1 (GABA-A Receptor)
GABRA1
Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.
Função
Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.
Medicamentos que Atuam neste Alvo
| Medicamento | Ação | Primário |
|---|---|---|
| Diazepam | Agonist | Sim |
| Alprazolam | Agonist | Sim |
| Zolpidem | Agonist | Sim |
| Memantine | Antagonist | Sim |
| Valproic Acid | Agonist | — |
| Topiramate | Agonist | — |