GABRA1 (GABA-A Receptor)

GABRA1

Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.

Функция

Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.

Препараты, действующие на данную мишень

Препарат Действие Первичный
Diazepam Agonist Да
Alprazolam Agonist Да
Zolpidem Agonist Да
Memantine Antagonist Да
Valproic Acid Agonist
Topiramate Agonist

Related Targets