SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
Функция
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
Препараты, действующие на данную мишень
| Препарат | Действие | Первичный |
|---|---|---|
| Valproic Acid | Blocker | Да |
| Topiramate | Blocker | Да |
| Phenytoin | Blocker | Да |
| Gabapentin | Blocker | Да |
| Pregabalin | Blocker | Да |
| Lamotrigine | Blocker | Да |
| Carbamazepine | Blocker | Да |
| Furosemide | Inhibitor | Да |
| Hydrochlorothiazide | Inhibitor | Да |