SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
İşlev
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
Bu Hedefe Etki Eden İlaçlar
| İlaç | Etki | Birincil |
|---|---|---|
| Valproic Acid | Blocker | Evet |
| Topiramate | Blocker | Evet |
| Phenytoin | Blocker | Evet |
| Gabapentin | Blocker | Evet |
| Pregabalin | Blocker | Evet |
| Lamotrigine | Blocker | Evet |
| Carbamazepine | Blocker | Evet |
| Furosemide | Inhibitor | Evet |
| Hydrochlorothiazide | Inhibitor | Evet |