SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
Fonction
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
Médicaments agissant sur cette cible
| Médicament | Action | Principal |
|---|---|---|
| Valproic Acid | Blocker | Oui |
| Topiramate | Blocker | Oui |
| Phenytoin | Blocker | Oui |
| Gabapentin | Blocker | Oui |
| Pregabalin | Blocker | Oui |
| Lamotrigine | Blocker | Oui |
| Carbamazepine | Blocker | Oui |
| Furosemide | Inhibitor | Oui |
| Hydrochlorothiazide | Inhibitor | Oui |