PDE5A (Phosphodiesterase 5)
PDE5A
cGMP-specific phosphodiesterase highly expressed in corpus cavernosum and pulmonary vasculature.
Função
PDE5 inhibitors (sildenafil, tadalafil) sustain cGMP signaling for erectile dysfunction and pulmonary arterial hypertension.
Medicamentos que Atuam neste Alvo
| Medicamento | Ação | Primário |
|---|---|---|
| Sildenafil | Inhibitor | Sim |
| Nitroglycerin | Other | Sim |