PDE5A (Phosphodiesterase 5)
PDE5A
cGMP-specific phosphodiesterase highly expressed in corpus cavernosum and pulmonary vasculature.
Fonction
PDE5 inhibitors (sildenafil, tadalafil) sustain cGMP signaling for erectile dysfunction and pulmonary arterial hypertension.
Médicaments agissant sur cette cible
| Médicament | Action | Principal |
|---|---|---|
| Sildenafil | Inhibitor | Oui |
| Nitroglycerin | Other | Oui |