PDE5A (Phosphodiesterase 5)
PDE5A
cGMP-specific phosphodiesterase highly expressed in corpus cavernosum and pulmonary vasculature.
Функция
PDE5 inhibitors (sildenafil, tadalafil) sustain cGMP signaling for erectile dysfunction and pulmonary arterial hypertension.
Препараты, действующие на данную мишень
| Препарат | Действие | Первичный |
|---|---|---|
| Sildenafil | Inhibitor | Да |
| Nitroglycerin | Other | Да |