PDE5A (Phosphodiesterase 5)
PDE5A
cGMP-specific phosphodiesterase highly expressed in corpus cavernosum and pulmonary vasculature.
Funktion
PDE5 inhibitors (sildenafil, tadalafil) sustain cGMP signaling for erectile dysfunction and pulmonary arterial hypertension.
Arzneimittel, die auf dieses Target wirken
| Arzneimittel | Wirkung | Primär |
|---|---|---|
| Sildenafil | Inhibitor | Ja |
| Nitroglycerin | Other | Ja |