SLC6A4 (Serotonin Transporter)

SLC6A4

Sodium-dependent serotonin transporter responsible for reuptake of 5-HT from the synaptic cleft.

Função

Primary target for SSRIs and SNRIs. Inhibition increases synaptic serotonin.

Medicamentos que Atuam neste Alvo

Medicamento Ação Primário
Sertraline Inhibitor Sim
Escitalopram Inhibitor Sim
Fluoxetine Inhibitor Sim
Duloxetine Inhibitor Sim
Venlafaxine Inhibitor Sim
Tramadol Inhibitor Sim
Ondansetron Other Sim
Quetiapine Inhibitor
Bupropion Inhibitor
Trazodone Inhibitor
Sumatriptan Other
Aripiprazole Partial Agonist

Related Targets