Procaine
A local anesthetic used to numb a specific area of the body during minor surgical procedures, dental work, or to relieve localized pain by temporarily blocking nerve signals. It was one of the first synthetic local anesthetics developed and has largely been replaced by longer-acting alternatives like lidocaine in most settings.
Peso Molecular
236,3100 g/mol
LogP
1,90
TPSA
55,60 Ų
Regra dos 5 de Lipinski
Aprovado
Áreas Terapêuticas
Mecanismo de Ação
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
Estrutura 2D
Cite this structure
Embed this structure
SMILES
CCN(CC)CCOC(=O)c1ccc(N)cc1
InChI
InChI=1S/C13H20N2O2/c1-3-15(4-2)9-10-17-13(16)11-5-7-12(14)8-6-11/h5-8H,3-4,9-10,14H2,1-2H3
Molecular Formula
C13H20N2O2
HBD / HBA
1 / 4
Ligações Rotacionáveis
7
Átomos Pesados
17
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Perguntas frequentes
A local anesthetic used to numb a specific area of the body during minor surgical procedures, dental work, or to relieve localized pain by temporarily blocking nerve signals. It was one of the first synthetic local anesthetics developed and has largely been replaced by longer-acting alternatives like lidocaine in most settings.
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
Yes, Procaine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL569. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 4914. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.
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