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Atenolol

CHEMBL24 Phase 4 Одобрено Small molecule
Half-Life
6-7 hours
Bioavailability
—
Protein Binding
—
Molecular Weight
266.3 g/mol
LogP
0.2
Phase
4

A beta-1 selective adrenergic blocker that slows the heart rate and reduces the force of heart contractions, lowering blood pressure and decreasing the heart's oxygen demand. It is used for hypertension, angina, and heart rhythm disorders including atrial fibrillation.

Молекулярная масса

266,3360 g/mol

LogP

0,20

TPSA

84,60 Ų

Правило пяти Липинского

Соответствует

Терапевтические области

Ovarian Cancer Pancreatic Cancer Bladder Cancer Thyroid Cancer Cardiovascular Disease Non-Small Cell Lung Cancer Osteoporosis Migraine Schizophrenia Chronic Kidney Disease Stroke Obesity Type 2 Diabetes Hypertension Breast Cancer Heart Failure Atrial Fibrillation Prostate Cancer Colorectal Cancer

Классы препаратов

C — C - Cardiovascular System

Механизм действия

Cardioselective beta-1 adrenergic receptor blocker without intrinsic sympathomimetic activity.

Pharmacokinetics (PK)

Half-Life 6-7 hours

Pharmacodynamics (PD)

Механизм

Cardioselective beta-1 adrenergic receptor blocker without intrinsic sympathomimetic activity.

2D Структура

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
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SMILES

                    
CC(C)NCC(O)COc1ccc(CC(N)=O)cc1

                

                

                
                

                    
InChI

                    
InChI=1S/C14H22N2O3/c1-10(2)16-8-12(17)9-19-13-5-3-11(4-6-13)7-14(15)18/h3-6,10,12,16-17H,7-9H2,1-2H3,(H2,15,18)

                

                

                

                    
                    

                        
Molecular Formula

                        
C14H22N2O3

                    

                    
                    

                        
HBD / HBA

                        
3 / 4

                    

                    
                    

                        
Вращаемые Связи

                        
8

                    

                    
                    
                    

                        
Тяжёлые Атомы

                        
19

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
Часто задаваемые вопросы

                

                    
                    

                        
                        

                            
A beta-1 selective adrenergic blocker that slows the heart rate and reduces the force of heart contractions, lowering blood pressure and decreasing the heart's oxygen demand. It is used for hypertension, angina, and heart rhythm disorders including atrial fibrillation.

                        

                    

                    

                    

                    
                    

                        
                        

                            
Cardioselective beta-1 adrenergic receptor blocker without intrinsic sympathomimetic activity.

                        

                    

                    

                    
                    

                        
                        

                            
Key pharmacokinetic parameters for Atenolol: Half-life: 6-7 hours.

                        

                    

                    

                    

                        
                        

                            
Yes, Atenolol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            
            

                
Related Drugs


                
                

                    
Same Drug Class

                    

                        
                        
                            Atorvastatin
                            Small molecule
                        
                        
                        
                            Amlodipine
                            Small molecule
                        
                        
                        
                            Lisinopril
                            Small molecule
                        
                        
                        
                            Metoprolol
                            Small molecule
                        
                        
                    

                

                

                
            

            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
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                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL24.
                Open-access bioactivity database.
            
        
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  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 2249.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.




        


        
        
    


    



    
Медицинский отказ от ответственности

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.