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Cangrelor

CHEMBL334966 Phase 4 Одобрено Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
776.4 g/mol
LogP
-1.0
Phase
4

A short-acting intravenous antiplatelet drug that rapidly inhibits the P2Y12 receptor to prevent platelet aggregation during and after heart procedures such as percutaneous coronary intervention. Its very short half-life allows quick reversal of antiplatelet effects, which is useful when bridging to oral therapy. It is used in patients who have not been pre-treated with oral P2Y12 inhibitors.

Молекулярная масса

776,4000 g/mol

LogP

-1,00

TPSA

307,00 Ų

Правило пяти Липинского

Не соответствует

Терапевтические области

Systemic Lupus Erythematosus Stroke

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D Структура

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
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SMILES

                    
CSCCNc1nc(SCCC(F)(F)F)nc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)C(Cl)(Cl)P(=O)(O)O)[C@@H](O)[C@H]1O

                

                

                
                

                    
InChI

                    
InChI=1S/C17H25Cl2F3N5O12P3S2/c1-43-5-3-23-12-9-13(26-15(25-12)44-4-2-16(20,21)22)27(7-24-9)14-11(29)10(28)8(38-14)6-37-42(35,36)39-41(33,34)17(18,19)40(30,31)32/h7-8,10-11,14,28-29H,2-6H2,1H3,(H,33,34)(H,35,36)(H,23,25,26)(H2,30,31,32)/t8-,10-,11-,14-/m1/s1

                

                

                

                    
                    

                        
Molecular Formula

                        
C17H25Cl2F3N5O12P3S2

                    

                    
                    

                        
HBD / HBA

                        
7 / 21

                    

                    
                    

                        
Вращаемые Связи

                        
15

                    

                    
                    
                    

                        
Тяжёлые Атомы

                        
44

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
Часто задаваемые вопросы

                

                    
                    

                        
                        

                            
A short-acting intravenous antiplatelet drug that rapidly inhibits the P2Y12 receptor to prevent platelet aggregation during and after heart procedures such as percutaneous coronary intervention. Its very short half-life allows quick reversal of antiplatelet effects, which is useful when bridging to oral therapy. It is used in patients who have not been pre-treated with oral P2Y12 inhibitors.

                        

                    

                    

                    

                    

                    

                    

                        
                        

                            
Yes, Cangrelor is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
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                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL334966.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 9854012.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.




        


        
        
    


    



    
Медицинский отказ от ответственности

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.