Copper Oxodotreotide

CHEMBL4302413 Phase 4 Đã phê duyệt Protein
Half-Life
Bioavailability
Protein Binding
Molecular Weight
g/mol
LogP
Phase
4

A copper-labeled form of a somatostatin analog used to target tumors that express somatostatin receptors, such as certain prostate cancers. It delivers therapeutic or diagnostic payloads directly to cancer cells.

Lĩnh vực điều trị

Cơ chế tác dụng

Competitively inhibits HMG-CoA reductase, the rate-limiting enzyme in the mevalonate pathway of cholesterol biosynthesis. This reduces intracellular cholesterol, upregulates LDL receptor expression, and lowers circulating LDL cholesterol.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Cơ chế

Competitively inhibits HMG-CoA reductase, the rate-limiting enzyme in the mevalonate pathway of cholesterol biosynthesis. This reduces intracellular cholesterol, upregulates LDL receptor expression, and lowers circulating LDL cholesterol.

HBD / HBA

- / -

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Câu hỏi thường gặp

A copper-labeled form of a somatostatin analog used to target tumors that express somatostatin receptors, such as certain prostate cancers. It delivers therapeutic or diagnostic payloads directly to cancer cells.

Competitively inhibits HMG-CoA reductase, the rate-limiting enzyme in the mevalonate pathway of cholesterol biosynthesis. This reduces intracellular cholesterol, upregulates LDL receptor expression, and lowers circulating LDL cholesterol.

Yes, Copper Oxodotreotide is an approved drug. It has reached clinical phase 4. It is classified as a Protein.

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References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL4302413. Open-access bioactivity database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-02-27.

Tuyên bố miễn trách y tế

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.