Pyrovalerone
Pyrovalerone is a psychostimulant cathinone derivative that inhibits the reuptake of dopamine and norepinephrine by blocking their respective monoamine transporters, producing CNS stimulation, increased alertness, and euphoria similar to cocaine. It was briefly investigated as a treatment for fatigue and lethargy but is now a controlled substance due to its significant abuse potential.
Khối lượng phân tử
245,3600 g/mol
LogP
3,80
TPSA
20,30 Ų
Lipinski RO5
Đạt
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Cấu trúc 2D
Cite this structure
Embed this structure
SMILES
CCCC(C(=O)c1ccc(C)cc1)N1CCCC1
InChI
InChI=1S/C16H23NO/c1-3-6-15(17-11-4-5-12-17)16(18)14-9-7-13(2)8-10-14/h7-10,15H,3-6,11-12H2,1-2H3
Molecular Formula
C16H23NO
HBD / HBA
- / 2
Liên kết có thể quay
5
Nguyên tử nặng
18
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Câu hỏi thường gặp
Pyrovalerone is a psychostimulant cathinone derivative that inhibits the reuptake of dopamine and norepinephrine by blocking their respective monoamine transporters, producing CNS stimulation, increased alertness, and euphoria similar to cocaine. It was briefly investigated as a treatment for fatigue and lethargy but is now a controlled substance due to its significant abuse potential.
Yes, Pyrovalerone is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL201960. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 14373. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.
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