Tetracaine

CHEMBL698 Phase 4 Đã phê duyệt Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
264.4 g/mol
LogP
3.7
Phase
4

This local anesthetic is used to numb specific areas of the body before medical procedures, and is commonly used as eye drops before eye examinations or minor eye surgery, as well as in spinal anesthesia. It works by blocking nerve signals in the targeted area to prevent pain sensation. It acts more slowly but longer than some other local anesthetics.

Khối lượng phân tử

264,3600 g/mol

LogP

3,70

TPSA

41,60 Ų

Lipinski RO5

Đạt

Lĩnh vực điều trị

Cơ chế tác dụng

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Cơ chế

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Cấu trúc 2D

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SMILES

CCCCNc1ccc(C(=O)OCCN(C)C)cc1

InChI

InChI=1S/C15H24N2O2/c1-4-5-10-16-14-8-6-13(7-9-14)15(18)19-12-11-17(2)3/h6-9,16H,4-5,10-12H2,1-3H3

Molecular Formula

C15H24N2O2

HBD / HBA

1 / 4

Liên kết có thể quay

9

Nguyên tử nặng

19

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Câu hỏi thường gặp

This local anesthetic is used to numb specific areas of the body before medical procedures, and is commonly used as eye drops before eye examinations or minor eye surgery, as well as in spinal anesthesia. It works by blocking nerve signals in the targeted area to prevent pain sensation. It acts more slowly but longer than some other local anesthetics.

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Yes, Tetracaine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL698. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 5411. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

Tuyên bố miễn trách y tế

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.