Labetalol

CHEMBL429 Phase 4 已批准 Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

328.4 g/mol

LogP

3.1

Phase

4

A combined alpha and beta-adrenergic blocker used to treat high blood pressure and hypertensive emergencies, including during pregnancy. It lowers blood pressure by reducing heart rate and relaxing blood vessels simultaneously.

分子量

328.4000 g/mol

LogP

3.10

TPSA

95.60 Å²

Lipinski 五规则

符合

治疗领域

Pain Management Asthma Epilepsy Migraine Schizophrenia Bipolar Disorder Generalized Anxiety Disorder Insomnia Chronic Kidney Disease Stroke Obesity Hypertension Chronic Pain Heart Failure

Pharmacokinetics (PK)

Pharmacodynamics (PD)

二维结构

SVG PNG

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SMILES

CC(CCc1ccccc1)NCC(O)c1ccc(O)c(C(N)=O)c1

InChI

InChI=1S/C19H24N2O3/c1-13(7-8-14-5-3-2-4-6-14)21-12-18(23)15-9-10-17(22)16(11-15)19(20)24/h2-6,9-11,13,18,21-23H,7-8,12H2,1H3,(H2,20,24)

Molecular Formula

C19H24N2O3

HBD / HBA

4 / 4

可旋转键数

8

重原子数

24

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

常见问题

A combined alpha and beta-adrenergic blocker used to treat high blood pressure and hypertensive emergencies, including during pregnancy. It lowers blood pressure by reducing heart rate and relaxing blood vessels simultaneously.

Yes, Labetalol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL429. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 3869. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

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结构

快速数据

分子式: C19H24N2O3
同义词: 4

外部链接

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医疗免责声明

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.