Bazedoxifene

CHEMBL46740 Phase 4 Approved Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

470.6 g/mol

LogP

6.1

Phase

4

A selective estrogen receptor modulator that acts as an estrogen antagonist in breast and uterine tissue while providing estrogen-like protection to bone, used to prevent postmenopausal osteoporosis.

Molecular Weight

470.6000 g/mol

LogP

6.10

TPSA

57.90 Å²

Lipinski RO5

Pass

Therapeutic Areas

Breast Cancer Endometriosis Generalized Anxiety Disorder Multiple Sclerosis Obesity Osteoporosis Schizophrenia

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D Structure

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SMILES

Cc1c(-c2ccc(O)cc2)n(Cc2ccc(OCCN3CCCCCC3)cc2)c2ccc(O)cc12

InChI

InChI=1S/C30H34N2O3/c1-22-28-20-26(34)12-15-29(28)32(30(22)24-8-10-25(33)11-9-24)21-23-6-13-27(14-7-23)35-19-18-31-16-4-2-3-5-17-31/h6-15,20,33-34H,2-5,16-19,21H2,1H3

Molecular Formula

C30H34N2O3

HBD / HBA

2 / 4

Rotatable Bonds

7

Heavy Atoms

35

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Frequently Asked Questions

A selective estrogen receptor modulator that acts as an estrogen antagonist in breast and uterine tissue while providing estrogen-like protection to bone, used to prevent postmenopausal osteoporosis.

Yes, Bazedoxifene is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL46740. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 154257. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

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Structure

Quick Data

Formula: C30H34N2O3

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Medical Disclaimer

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.