ADRB1 (Beta-1 Adrenergic Receptor)

ADRB1

G-protein coupled receptor (Gs) predominantly expressed in the heart.

Fonction

Beta-1 selective blockers (metoprolol, bisoprolol) treat hypertension, heart failure, and arrhythmias.

Médicaments agissant sur cette cible

Médicament Action Principal
Carvedilol Antagonist Oui
Metoprolol Antagonist Oui
Propranolol Antagonist Oui
Albuterol Agonist

Related Targets