ADRB1 (Beta-1 Adrenergic Receptor)

ADRB1

G-protein coupled receptor (Gs) predominantly expressed in the heart.

Fonction

Beta-1 selective blockers (metoprolol, bisoprolol) treat hypertension, heart failure, and arrhythmias.

Médicaments agissant sur cette cible

Médicament Action Principal
Carvedilol Antagonist Oui
Metoprolol Antagonist Oui
Propranolol Antagonist Oui
Albuterol Agonist —

Related Targets