OPRM1 (Mu-Opioid Receptor)

OPRM1

G-protein coupled receptor (Gi/o) mediating analgesia, euphoria, respiratory depression, and physical dependence.

Fonction

Primary target for opioid analgesics (morphine, fentanyl, oxycodone). Activation produces potent analgesia but also respiratory depression and addiction.

Médicaments agissant sur cette cible

Médicament Action Principal
Morphine Agonist Oui
Oxycodone Agonist Oui
Tramadol Agonist

Related Targets