Carbamoylcholine

CHEMBL965 Phase 4 承認済み Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
147.2 g/mol
LogP
-0.4
Phase
4

Another name for carbachol, a cholinomimetic agent that activates both muscarinic and nicotinic acetylcholine receptors. It is used as an ophthalmic agent to constrict the pupil and lower intraocular pressure. It is resistant to cholinesterase-mediated breakdown, resulting in a prolonged duration of action.

分子量

147.2000 g/mol

LogP

-0.40

TPSA

52.30 Ų

リピンスキーの五則

適合

作用機序

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

機序

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

2D構造

SVG PNG

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SMILES

C[N+](C)(C)CCOC(N)=O

InChI

InChI=1S/C6H14N2O2/c1-8(2,3)4-5-10-6(7)9/h4-5H2,1-3H3,(H-,7,9)/p+1

Molecular Formula

C6H15N2O2+

HBD / HBA

1 / 2

回転可能結合数

4

重原子数

10

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

よくある質問

Another name for carbachol, a cholinomimetic agent that activates both muscarinic and nicotinic acetylcholine receptors. It is used as an ophthalmic agent to constrict the pupil and lower intraocular pressure. It is resistant to cholinesterase-mediated breakdown, resulting in a prolonged duration of action.

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Yes, Carbamoylcholine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL965. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 2551. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

医学的免責事項

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.