HRH1 (Histamine H1 Receptor)

HRH1

G-protein coupled receptor (Gq) mediating allergic and inflammatory responses.

機能

H1 antagonists (antihistamines) block histamine-induced vasodilation, itching, and bronchoconstriction.

この標的に作用する薬物

薬物 作用 主要
Cetirizine Antagonist はい
Diphenhydramine Antagonist はい
Loratadine Antagonist はい
Quetiapine Antagonist
Trazodone Antagonist

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