HRH1 (Histamine H1 Receptor)

HRH1

G-protein coupled receptor (Gq) mediating allergic and inflammatory responses.

Функция

H1 antagonists (antihistamines) block histamine-induced vasodilation, itching, and bronchoconstriction.

Препараты, действующие на данную мишень

Препарат Действие Первичный
Cetirizine Antagonist Да
Diphenhydramine Antagonist Да
Loratadine Antagonist Да
Quetiapine Antagonist
Trazodone Antagonist

Related Targets