EGFR (Epidermal Growth Factor Receptor)

EGFR

Receptor tyrosine kinase driving cell proliferation, commonly mutated in NSCLC.

Function

Activating mutations drive oncogenic signaling. Targeted by TKIs (erlotinib, osimertinib) and antibodies (cetuximab).

Drugs Acting on This Target

Drug Action Primary
Trastuzumab Antagonist Yes

Related Targets