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Pyrilamine

CHEMBL511 Phase 4 ได้รับการอนุมัติ Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
285.4 g/mol
LogP
3.3
Phase
4

Pyrilamine is a first-generation antihistamine of the ethylenediamine class that competitively antagonizes histamine H1 receptors, reducing allergic symptoms including rhinorrhea, sneezing, and pruritus, and also possesses significant anticholinergic and sedative properties. It is used in combination over-the-counter products for allergy, cold, and sleep aid formulations.

น้ำหนักโมเลกุล

285.4000 g/mol

LogP

3.30

TPSA

28.60 Ų

Lipinski RO5

ผ่าน

Pharmacokinetics (PK)

Pharmacodynamics (PD)

โครงสร้าง 2 มิติ

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
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SMILES

                    
COc1ccc(CN(CCN(C)C)c2ccccn2)cc1

                

                

                
                

                    
InChI

                    
InChI=1S/C17H23N3O/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15/h4-11H,12-14H2,1-3H3

                

                

                

                    
                    

                        
Molecular Formula

                        
C17H23N3O

                    

                    
                    

                        
HBD / HBA

                        
- / 4

                    

                    
                    

                        
พันธะที่หมุนได้

                        
7

                    

                    
                    
                    

                        
อะตอมหนัก

                        
21

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
คำถามที่พบบ่อย

                

                    
                    

                        
                        

                            
Pyrilamine is a first-generation antihistamine of the ethylenediamine class that competitively antagonizes histamine H1 receptors, reducing allergic symptoms including rhinorrhea, sneezing, and pruritus, and also possesses significant anticholinergic and sedative properties. It is used in combination over-the-counter products for allergy, cold, and sleep aid formulations.

                        

                    

                    

                    

                    

                    

                    

                        
                        

                            
Yes, Pyrilamine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
  • 
            
            
                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL511.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 4992.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.




        


        
        
    


    



    
ข้อจำกัดความรับผิดชอบทางการแพทย์

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.