Cyproheptadine Hydrochloride
The hydrochloride salt of cyproheptadine, an antihistamine with antiserotonin effects used for allergic conditions and appetite stimulation. It causes sedation and may be used as a sleep aid in some patients.
分子量
323.9000 g/mol
TPSA
3.20 Ų
治疗领域
作用机制
Competitively blocks histamine H1 receptors on effector cells, preventing histamine-mediated vasodilation, increased vascular permeability, bronchoconstriction, and pruritus. First-generation agents also cross the blood-brain barrier, causing sedation.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Competitively blocks histamine H1 receptors on effector cells, preventing histamine-mediated vasodilation, increased vascular permeability, bronchoconstriction, and pruritus. First-generation agents also cross the blood-brain barrier, causing sedation.
二维结构
Cite this structure
Embed this structure
SMILES
CN1CCC(=C2c3ccccc3C=Cc3ccccc32)CC1.Cl
InChI
InChI=1S/C21H21N.ClH/c1-22-14-12-18(13-15-22)21-19-8-4-2-6-16(19)10-11-17-7-3-5-9-20(17)21;/h2-11H,12-15H2,1H3;1H
Molecular Formula
C21H22ClN
HBD / HBA
1 / 1
可旋转键数
0
重原子数
23
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
常见问题
The hydrochloride salt of cyproheptadine, an antihistamine with antiserotonin effects used for allergic conditions and appetite stimulation. It causes sedation and may be used as a sleep aid in some patients.
Competitively blocks histamine H1 receptors on effector cells, preventing histamine-mediated vasodilation, increased vascular permeability, bronchoconstriction, and pruritus. First-generation agents also cross the blood-brain barrier, causing sedation.
Yes, Cyproheptadine Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1716. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 13770. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.
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