Fentanyl
This is a potent opioid pain reliever that works by binding to opioid receptors in the brain and spinal cord to block pain signals. Due to its high potency, it carries significant risks of dependence and overdose and requires careful medical supervision.
Molekularmasse
336,4700 g/mol
LogP
4,00
TPSA
23,60 Ų
Lipinski-Regel der Fünf
Bestanden
Therapeutische Bereiche
Arzneimittelklassen
Wirkmechanismus
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
2D-Struktur
Cite this structure
Embed this structure
SMILES
CCC(=O)N(c1ccccc1)C1CCN(CCc2ccccc2)CC1
InChI
InChI=1S/C22H28N2O/c1-2-22(25)24(20-11-7-4-8-12-20)21-14-17-23(18-15-21)16-13-19-9-5-3-6-10-19/h3-12,21H,2,13-18H2,1H3
Molecular Formula
C22H28N2O
HBD / HBA
- / 2
Rotierbare Bindungen
6
Schwere Atome
25
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Häufig gestellte Fragen
This is a potent opioid pain reliever that works by binding to opioid receptors in the brain and spinal cord to block pain signals. Due to its high potency, it carries significant risks of dependence and overdose and requires careful medical supervision.
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
Key pharmacokinetic parameters for Fentanyl: Half-life: 2-4 hours.
Yes, Fentanyl is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
Related Drugs
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL596. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 3345. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.
Medizinischer Haftungsausschluss
This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
Embed This Widget
Add the script tag and a data attribute to embed this widget.
<script src="https://cdn.jsdelivr.net/npm/drugfyi-embed@1/dist/embed.min.js" defer></script>
<div data-drugfyi="drug" data-slug="fentanyl"></div>Embed via iframe for maximum compatibility.
<iframe src="https://drugfyi.com/iframe/drug/fentanyl/" width="420" height="400" frameborder="0" style="border:0;border-radius:10px;max-width:100%" loading="lazy"></iframe>Paste this URL in WordPress, Medium, or any oEmbed-compatible platform.
https://drugfyi.com/drug/fentanyl/Add a dynamic SVG badge to your README or docs.
[](https://drugfyi.com/drug/fentanyl/)Use the native HTML custom element.
<script src="https://cdn.jsdelivr.net/npm/drugfyi-embed@1/dist/embed.min.js" defer></script>
<drugfyi-drug slug="fentanyl"></drugfyi-drug>