Fentanyl
This is a potent opioid pain reliever that works by binding to opioid receptors in the brain and spinal cord to block pain signals. Due to its high potency, it carries significant risks of dependence and overdose and requires careful medical supervision.
Peso Molecular
336,4700 g/mol
LogP
4,00
TPSA
23,60 Ų
Regra dos 5 de Lipinski
Aprovado
Áreas Terapêuticas
Classes de Medicamentos
Mecanismo de Ação
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
Estrutura 2D
Cite this structure
Embed this structure
SMILES
CCC(=O)N(c1ccccc1)C1CCN(CCc2ccccc2)CC1
InChI
InChI=1S/C22H28N2O/c1-2-22(25)24(20-11-7-4-8-12-20)21-14-17-23(18-15-21)16-13-19-9-5-3-6-10-19/h3-12,21H,2,13-18H2,1H3
Molecular Formula
C22H28N2O
HBD / HBA
- / 2
Ligações Rotacionáveis
6
Átomos Pesados
25
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Perguntas frequentes
This is a potent opioid pain reliever that works by binding to opioid receptors in the brain and spinal cord to block pain signals. Due to its high potency, it carries significant risks of dependence and overdose and requires careful medical supervision.
Highly potent synthetic mu-opioid receptor agonist approximately 100 times more potent than morphine.
Key pharmacokinetic parameters for Fentanyl: Half-life: 2-4 hours.
Yes, Fentanyl is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
Related Drugs
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL596. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 3345. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.
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