Labetalol

CHEMBL429 Phase 4 Aprovado Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

328.4 g/mol

LogP

3.1

Phase

4

A combined alpha and beta-adrenergic blocker used to treat high blood pressure and hypertensive emergencies, including during pregnancy. It lowers blood pressure by reducing heart rate and relaxing blood vessels simultaneously.

Peso Molecular

328,4000 g/mol

LogP

3,10

TPSA

95,60 Å²

Regra dos 5 de Lipinski

Aprovado

Áreas Terapêuticas

Pain Management Asthma Epilepsy Migraine Schizophrenia Bipolar Disorder Generalized Anxiety Disorder Insomnia Chronic Kidney Disease Stroke Obesity Hypertension Chronic Pain Heart Failure

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Estrutura 2D

SVG PNG

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SMILES

CC(CCc1ccccc1)NCC(O)c1ccc(O)c(C(N)=O)c1

InChI

InChI=1S/C19H24N2O3/c1-13(7-8-14-5-3-2-4-6-14)21-12-18(23)15-9-10-17(22)16(11-15)19(20)24/h2-6,9-11,13,18,21-23H,7-8,12H2,1H3,(H2,20,24)

Molecular Formula

C19H24N2O3

HBD / HBA

4 / 4

Ligações Rotacionáveis

8

Átomos Pesados

24

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Perguntas frequentes

A combined alpha and beta-adrenergic blocker used to treat high blood pressure and hypertensive emergencies, including during pregnancy. It lowers blood pressure by reducing heart rate and relaxing blood vessels simultaneously.

Yes, Labetalol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL429. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 3869. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

PillFYI

Procura informações acessíveis para o paciente?

Labetalol no PillFYI

Estrutura

Dados Rápidos

Fórmula: C19H24N2O3
Sinônimos: 4

Links Externos

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Aviso Médico

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.