Tapentadol

CHEMBL1201776 Phase 4 Onaylandı Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

221.3 g/mol

LogP

3.5

Phase

4

This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

Moleküler Ağırlık

221,3400 g/mol

LogP

3,50

TPSA

23,50 Å²

Lipinski RO5

Geçer

Terapötik Alanlar

Ovarian Cancer Pancreatic Cancer Bladder Cancer Thyroid Cancer Pain Management Non-Small Cell Lung Cancer Rheumatoid Arthritis Breast Cancer Chronic Pain Prostate Cancer Colorectal Cancer

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D Yapı

SVG PNG

Cite this structure

Embed this structure

SMILES

CC[C@@H](c1cccc(O)c1)[C@@H](C)CN(C)C

InChI

InChI=1S/C14H23NO/c1-5-14(11(2)10-15(3)4)12-7-6-8-13(16)9-12/h6-9,11,14,16H,5,10H2,1-4H3/t11-,14+/m0/s1

Molecular Formula

C14H23NO

HBD / HBA

1 / 2

Döndürülebilir Bağlar

5

Ağır Atomlar

16

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

Yes, Tapentadol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201776. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 9838022. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

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Hızlı Veriler

Formül: C14H23NO
Eş Anlamlılar: 2

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This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.