Prodrug
A pharmacologically inactive compound that is metabolically converted to an active drug in vivo. Used to improve bioavailability, reduce toxicity, or target specific tissues.
Ví dụ
- Enalapril -> enalaprilat
- Codeine -> morphine (CYP2D6)
- Valacyclovir -> acyclovir
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A pharmacologically inactive compound that is metabolically converted to an active drug in vivo. Used to improve bioavailability, reduce toxicity, or target specific tissues.