HRH1 (Histamine H1 Receptor)

HRH1

G-protein coupled receptor (Gq) mediating allergic and inflammatory responses.

功能

H1 antagonists (antihistamines) block histamine-induced vasodilation, itching, and bronchoconstriction.

作用于该靶点的药物

药物 作用 主要
Trazodone Antagonist
Cetirizine Antagonist
Loratadine Antagonist
Diphenhydramine Antagonist
Memantine Antagonist
Quetiapine Antagonist
Ondansetron Antagonist
Escitalopram Antagonist

Related Targets