HRH1 (Histamine H1 Receptor)

HRH1

G-protein coupled receptor (Gq) mediating allergic and inflammatory responses.

Fonction

H1 antagonists (antihistamines) block histamine-induced vasodilation, itching, and bronchoconstriction.

Médicaments agissant sur cette cible

Médicament Action Principal
Trazodone Antagonist Oui
Cetirizine Antagonist Oui
Loratadine Antagonist Oui
Diphenhydramine Antagonist Oui
Memantine Antagonist
Quetiapine Antagonist
Ondansetron Antagonist
Escitalopram Antagonist

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