HRH1 (Histamine H1 Receptor)

HRH1

G-protein coupled receptor (Gq) mediating allergic and inflammatory responses.

Fonction

H1 antagonists (antihistamines) block histamine-induced vasodilation, itching, and bronchoconstriction.

Médicaments agissant sur cette cible

Médicament Action Principal
Cetirizine Antagonist Oui
Diphenhydramine Antagonist Oui
Loratadine Antagonist Oui
Quetiapine Antagonist
Trazodone Antagonist

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