PPARG (Peroxisome Proliferator-Activated Receptor Gamma)
PPARG
Nuclear receptor regulating glucose and lipid metabolism, adipocyte differentiation.
功能
Thiazolidinediones (pioglitazone) activate PPARG to improve insulin sensitivity.
作用于该靶点的药物
| 药物 | 作用 | 主要 |
|---|---|---|
| Methylprednisolone | Agonist | 是 |
| Insulin Glargine | Agonist | 是 |
| Liraglutide | Agonist | 是 |
| Semaglutide | Agonist | 是 |
| Tirzepatide | Agonist | 是 |
| Prednisone | Agonist | 是 |
| Dexamethasone | Agonist | 是 |
| Levothyroxine | Agonist | 是 |
| Spironolactone | Antagonist | 是 |
| Tamoxifen | Antagonist | 是 |
| Sitagliptin | Inhibitor | 是 |
| Finasteride | Inhibitor | 是 |
| Empagliflozin | Inhibitor | 是 |
| Metformin | Other | 是 |
| Montelukast | Other | — |