ADRB2 (Beta-2 Adrenergic Receptor)

ADRB2

G-protein coupled receptor (Gs) expressed in bronchial smooth muscle and vasculature.

Function

Beta-2 agonists (albuterol, salmeterol) are first-line bronchodilators for asthma and COPD.

Drugs Acting on This Target

Drug Action Primary
Albuterol Agonist Yes
Carvedilol Antagonist
Propranolol Antagonist
Metoprolol Antagonist

Related Targets