AGTR1 (Angiotensin II Type 1 Receptor)

AGTR1

G-protein coupled receptor mediating vasoconstriction and aldosterone release.

Function

ARBs (losartan, valsartan) selectively block AT1, providing RAAS inhibition without ACE inhibitor cough.

Drugs Acting on This Target

Drug Action Primary
Losartan Antagonist Yes
Valsartan Antagonist Yes
Amlodipine Other Yes
Spironolactone Other

Related Targets