ADRB2 (Beta-2 Adrenergic Receptor)

ADRB2

G-protein coupled receptor (Gs) expressed in bronchial smooth muscle and vasculature.

Funktion

Beta-2 agonists (albuterol, salmeterol) are first-line bronchodilators for asthma and COPD.

Arzneimittel, die auf dieses Target wirken

Arzneimittel Wirkung Primär
Albuterol Agonist Ja
Sumatriptan Agonist Ja
Tamsulosin Antagonist Ja
Carvedilol Antagonist
Metoprolol Antagonist
Propranolol Antagonist
Amlodipine Other

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