DRD2 (Dopamine D2 Receptor)

DRD2

G-protein coupled receptor (Gi/o) mediating dopaminergic neurotransmission.

Funktion

Key target for antipsychotic drugs (antagonists) and anti-parkinsonian agents (agonists). D2 blockade in the mesolimbic pathway reduces positive psychotic symptoms.

Arzneimittel, die auf dieses Target wirken

Arzneimittel Wirkung Primär
Levodopa Agonist Ja
Quetiapine Antagonist Ja
Aripiprazole Partial Agonist Ja

Related Targets