DRD2 (Dopamine D2 Receptor)
DRD2
G-protein coupled receptor (Gi/o) mediating dopaminergic neurotransmission.
기능
Key target for antipsychotic drugs (antagonists) and anti-parkinsonian agents (agonists). D2 blockade in the mesolimbic pathway reduces positive psychotic symptoms.
이 표적에 작용하는 약물
| 약물 | 작용 | 주요 |
|---|---|---|
| Levodopa | Agonist | 예 |
| Quetiapine | Antagonist | 예 |
| Aripiprazole | Partial Agonist | 예 |
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SIGMAR1 (Sigma-1 Receptor)
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CTLA4 (Cytotoxic T-Lymphocyte Antigen 4)
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ADRB1 (Beta-1 Adrenergic Receptor)
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ADRB2 (Beta-2 Adrenergic Receptor)
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HRH2 (Histamine H2 Receptor)
HRH2